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Assay Detail

CHEMBL4330008

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of recombinant human CYP1A1 expressed in Escherichia coli membranes co-expressing NADPH-P450 reductase assessed as reduction in ethoxyresorufin O-de-ethylation preincubated for 3 mins followed by NADPH addition and measured after 10 mins by fluorometric method
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 1A1 (CHEMBL2231)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Adaptable Small Ligand of CYP1 Enzymes for Use in Understanding the Structural Features Determining Isoform Selectivity.
Lee JY, Cho H, Thangapandian S, Lim C, Chun YJ, Lee Y, Choi S, Kim S.
ACS Med Chem Lett (2018) 9 : 1247 -1252
PubMed 30613334 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 7.10 7.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4447260 1 7.39
CHEMBL283196 ALPHA-NAPHTHOFLAVONE 1 7.26
CHEMBL42428 1 7.21
CHEMBL46909 1 6.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4447260 IC50 = 41.0 nM 7.39
CHEMBL283196 ALPHA-NAPHTHOFLAVONE IC50 = 55.0 nM 7.26
CHEMBL42428 IC50 = 61.0 nM 7.21
CHEMBL46909 IC50 = 300.0 nM 6.52