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Assay Detail

CHEMBL4339724

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Antagonist activity at CCR5 (unknown origin) expressed in human HT1080 cells assessed as blockade of MIP1beta-binding to receptor
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

C-C chemokine receptor type 5 (CHEMBL274)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Use of a Conformational-Switching Mechanism to Modulate Exposed Polarity: Discovery of CCR2 Antagonist BMS-741672.
Yang MG, Xiao Z, Cherney RJ, Tebben AJ, Batt DG, Brown GD, Chen J, Cvijic ME, Dabros M, Duncia JV, Galella M, Gardner DS, Khandelwal P, Ko SS, Malley MF, Mo R, Pang J, Rose AV, Santella JB, Shi H, Srivastava A, Traeger SC, Wang B, Xu S, Zhao R, Barrish JC, Mandlekar S, Zhao Q, Carter PH.
ACS Med Chem Lett (2019) 10 : 300 -305
PubMed 30891130 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 6.43 8.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3577945 1 8.62
CHEMBL4470701 1 6.72
CHEMBL4457723 BMS-741672 2.0 1 6.54
CHEMBL4442783 1 6.11
CHEMBL4465351 1 5.80
CHEMBL3233178 1 5.79
CHEMBL4463290 1 5.46

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3577945 IC50 = 2.4 nM 8.62
CHEMBL4470701 IC50 = 190.0 nM 6.72
CHEMBL4457723 BMS-741672 IC50 = 287.0 nM 6.54
CHEMBL4442783 IC50 = 780.0 nM 6.11
CHEMBL4465351 IC50 = 1570.0 nM 5.80
CHEMBL3233178 IC50 = 1636.0 nM 5.79
CHEMBL4463290 IC50 = 3469.0 nM 5.46