Assay Detail
Binding
CHEMBL4346780
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant full length His-tagged CDK9/cyclin K expressed in baculovirus expression system
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Cyclin-Dependent Kinase 2 Inhibitors in Cancer Therapy: An Update.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.52 | 8.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1944698 | ZOTIRACICLIB | 2.0 | 1 | 8.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1944698 | ZOTIRACICLIB | IC50 | = | 3.0 | nM | 8.52 |