Assay Detail
Binding
CHEMBL4351061
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of DcpS (unknown origin) using m7GpppA as substrate by ELISA
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Emerging and Re-Emerging Warheads for Targeted Covalent Inhibitors: Applications in Medicinal Chemistry and Chemical Biology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.49 | 8.49 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL342595 | — | — | 1 | 8.49 |
| CHEMBL4465809 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL342595 | — | IC50 | = | 3.2 | nM | 8.49 |
| CHEMBL4465809 | — | IC50 | < | 0.02 | nM | - |