Assay Detail
Functional
CHEMBL4352819
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Enterovirus A71 infected in human RD cells assessed as reduction in virus-induced cell death incubated for 4 days by CellTiter-Glo luminescence assay
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Enterovirus A71 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design, synthesis and pharmacological evaluation of a novel mTOR-targeted anti-EV71 agent.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 31 | 6.23 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1765602 | — | — | 1 | 8.00 |
| CHEMBL4525212 | — | — | 1 | 7.57 |
| CHEMBL4453904 | — | — | 1 | 7.40 |
| CHEMBL4562378 | — | — | 1 | 7.23 |
| CHEMBL4573610 | — | — | 1 | 7.16 |
| CHEMBL4465800 | — | — | 1 | 7.05 |
| CHEMBL4459882 | — | — | 1 | 7.05 |
| CHEMBL4550789 | — | — | 1 | 6.77 |
| CHEMBL4580312 | — | — | 1 | 6.70 |
| CHEMBL4475823 | — | — | 1 | 6.57 |
| CHEMBL4459925 | — | — | 1 | 6.25 |
| CHEMBL4472012 | — | — | 1 | 6.09 |
| CHEMBL4459449 | — | — | 1 | 6.05 |
| CHEMBL4581200 | — | — | 1 | 5.61 |
| CHEMBL4466203 | — | — | 1 | 5.61 |
| CHEMBL4533872 | — | — | 1 | 5.61 |
| CHEMBL4447635 | — | — | 1 | 5.58 |
| CHEMBL4453652 | — | — | 1 | 5.32 |
| CHEMBL4447016 | — | — | 1 | 5.29 |
| CHEMBL4540379 | — | — | 1 | 5.13 |
| CHEMBL4472225 | — | — | 1 | 4.62 |
| CHEMBL4453549 | — | — | 1 | 4.31 |
| CHEMBL4562087 | — | — | 1 | - |
| CHEMBL4559116 | — | — | 1 | - |
| CHEMBL4436243 | — | — | 1 | - |
| CHEMBL4548073 | — | — | 1 | - |
| CHEMBL4576178 | — | — | 1 | - |
| CHEMBL4575223 | — | — | 1 | - |
| CHEMBL4577216 | — | — | 1 | - |
| CHEMBL4471220 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1765602 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4525212 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL4453904 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL4562378 | — | IC50 | = | 59.0 | nM | 7.23 |
| CHEMBL4573610 | — | IC50 | = | 70.0 | nM | 7.16 |
| CHEMBL4465800 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL4459882 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL4550789 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL4580312 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL4475823 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL4459925 | — | IC50 | = | 560.0 | nM | 6.25 |
| CHEMBL4472012 | — | IC50 | = | 820.0 | nM | 6.09 |
| CHEMBL4459449 | — | IC50 | = | 890.0 | nM | 6.05 |
| CHEMBL4581200 | — | IC50 | = | 2470.0 | nM | 5.61 |
| CHEMBL4533872 | — | IC50 | = | 2470.0 | nM | 5.61 |
| CHEMBL4466203 | — | IC50 | = | 2470.0 | nM | 5.61 |
| CHEMBL4447635 | — | IC50 | = | 2630.0 | nM | 5.58 |
| CHEMBL4453652 | — | IC50 | = | 4780.0 | nM | 5.32 |
| CHEMBL4447016 | — | IC50 | = | 5140.0 | nM | 5.29 |
| CHEMBL4540379 | — | IC50 | = | 7400.0 | nM | 5.13 |
| CHEMBL4472225 | — | IC50 | = | 23720.0 | nM | 4.62 |
| CHEMBL4453549 | — | IC50 | = | 48900.0 | nM | 4.31 |
| CHEMBL4518633 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4471220 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4577216 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4575223 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4576178 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4548073 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4436243 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4559116 | — | IC50 | > | 200000.0 | nM | - |
| CHEMBL4562087 | — | IC50 | > | 200000.0 | nM | - |