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Assay Detail

CHEMBL4354904

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Binding
Binding affinity to Streptococcus mutans Sortase A
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Streptococcus mutans
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sortase A (CHEMBL4523939)
Type SINGLE PROTEIN
Organism Streptococcus mutans

Publication

Targeting <i>S. mutans</i> biofilms: a perspective on preventing dental caries.
Scharnow AM, Solinski AE, Wuest WM.
Medchemcomm (2019) 10 : 1057 -1067
PubMed 31391878 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.95 5.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7976 CHALCONE 1 5.30
CHEMBL140 CURCUMIN 3.0 1 4.99
CHEMBL28626 MORIN 1 4.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7976 CHALCONE IC50 = 5000.0 nM 5.30
CHEMBL140 CURCUMIN IC50 = 10200.0 nM 4.99
CHEMBL28626 MORIN IC50 = 27200.0 nM 4.57