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Assay Detail

CHEMBL4355296

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Binding
Inhibition of Plasmodium falciparum plasmepsin 2 using fluorescently labeled peptide substrate by fluorescence method
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Plasmodium falciparum
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Plasmepsin II (CHEMBL4414)
Type SINGLE PROTEIN
Organism Plasmodium falciparum

Publication

Exploiting Structural Dynamics To Design Open-Flap Inhibitors of Malarial Aspartic Proteases.
Bobrovs R, Jaudzems K, Jirgensons A.
J Med Chem (2019) 62 : 8931 -8950
PubMed 31062983 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 15 6.38 7.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4456145 1 7.52
CHEMBL4585628 1 7.30
CHEMBL4578117 1 7.16
CHEMBL4541926 1 6.89
CHEMBL4552145 1 6.82
CHEMBL4457677 1 6.77
CHEMBL4436986 1 6.72
CHEMBL4553173 1 6.46
CHEMBL4456617 1 6.42
CHEMBL4472299 1 6.17
CHEMBL4554580 1 5.71
CHEMBL4590673 1 5.38
CHEMBL4581864 1 5.30
CHEMBL4558605 1 4.72
CHEMBL4442042 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4456145 IC50 = 30.0 nM 7.52
CHEMBL4585628 IC50 = 50.0 nM 7.30
CHEMBL4578117 IC50 = 70.0 nM 7.16
CHEMBL4541926 IC50 = 130.0 nM 6.89
CHEMBL4552145 IC50 = 150.0 nM 6.82
CHEMBL4457677 IC50 = 170.0 nM 6.77
CHEMBL4436986 IC50 = 190.0 nM 6.72
CHEMBL4553173 IC50 = 350.0 nM 6.46
CHEMBL4456617 IC50 = 380.0 nM 6.42
CHEMBL4472299 IC50 = 680.0 nM 6.17
CHEMBL4554580 IC50 = 1950.0 nM 5.71
CHEMBL4590673 IC50 = 4190.0 nM 5.38
CHEMBL4581864 IC50 = 5000.0 nM 5.30
CHEMBL4558605 IC50 = 19000.0 nM 4.72
CHEMBL4442042 IC50 <= 45.0 nM -