Assay Detail
Functional
CHEMBL4360799
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Antiviral activity against Human rhinovirus A2
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | rhinovirus A2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Back to the future: Advances in development of broad-spectrum capsid-binding inhibitors of enteroviruses.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 7.64 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL283639 | DISOXARIL | 2.0 | 1 | 8.40 |
| CHEMBL96339 | — | — | 1 | 8.05 |
| CHEMBL320168 | — | — | 1 | 8.05 |
| CHEMBL328858 | — | — | 1 | 8.05 |
| CHEMBL230440 | — | — | 1 | 8.05 |
| CHEMBL395062 | — | — | 1 | 8.05 |
| CHEMBL396266 | — | — | 1 | 8.05 |
| CHEMBL397439 | — | — | 1 | 8.05 |
| CHEMBL231280 | — | — | 1 | 8.05 |
| CHEMBL231378 | — | — | 1 | 8.05 |
| CHEMBL397440 | — | — | 1 | 8.05 |
| CHEMBL4541546 | — | — | 1 | 8.05 |
| CHEMBL4469987 | — | — | 1 | 7.40 |
| CHEMBL6641 | — | — | 1 | 7.40 |
| CHEMBL6824 | — | — | 1 | 7.40 |
| CHEMBL25488 | — | — | 1 | 7.00 |
| CHEMBL266800 | — | — | 1 | 7.00 |
| CHEMBL28442 | — | — | 1 | 6.05 |
| CHEMBL293278 | — | — | 1 | 6.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL283639 | DISOXARIL | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL96339 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL320168 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL328858 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL230440 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL395062 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL396266 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL397439 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL231280 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL231378 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL397440 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL4541546 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL4469987 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL6641 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL6824 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL25488 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL266800 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL28442 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL293278 | — | IC50 | = | 900.0 | nM | 6.05 |