Assay Detail
Binding
CHEMBL4375086
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Inhibition of Bcl-XL (unknown origin) by fluorescence polarization assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structure-Guided Discovery of a Selective Mcl-1 Inhibitor with Cellular Activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 15 | 4.56 | 4.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4460382 | — | — | 1 | 4.82 |
| CHEMBL4455822 | — | — | 1 | 4.77 |
| CHEMBL4472592 | — | — | 1 | 4.75 |
| CHEMBL4450255 | — | — | 1 | 4.75 |
| CHEMBL4514111 | — | — | 1 | 4.62 |
| CHEMBL4442085 | — | — | 1 | 4.58 |
| CHEMBL4573285 | — | — | 1 | 4.48 |
| CHEMBL4521569 | — | — | 1 | 4.41 |
| CHEMBL4443675 | — | — | 1 | 4.38 |
| CHEMBL4456249 | — | — | 1 | 4.06 |
| CHEMBL4440978 | — | — | 1 | - |
| CHEMBL4455139 | — | — | 1 | - |
| CHEMBL4471326 | — | — | 1 | - |
| CHEMBL4448439 | — | — | 1 | - |
| CHEMBL4436725 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4460382 | — | Ki | = | 15000.0 | nM | 4.82 |
| CHEMBL4455822 | — | Ki | = | 17000.0 | nM | 4.77 |
| CHEMBL4472592 | — | Ki | = | 18000.0 | nM | 4.75 |
| CHEMBL4450255 | — | Ki | = | 18000.0 | nM | 4.75 |
| CHEMBL4514111 | — | Ki | = | 24000.0 | nM | 4.62 |
| CHEMBL4442085 | — | Ki | = | 26000.0 | nM | 4.58 |
| CHEMBL4573285 | — | Ki | = | 33000.0 | nM | 4.48 |
| CHEMBL4521569 | — | Ki | = | 39000.0 | nM | 4.41 |
| CHEMBL4443675 | — | Ki | = | 42000.0 | nM | 4.38 |
| CHEMBL4456249 | — | Ki | = | 87000.0 | nM | 4.06 |
| CHEMBL4440978 | — | Ki | = | 216000.0 | nM | - |
| CHEMBL4455139 | — | Ki | = | 319000.0 | nM | - |
| CHEMBL4471326 | — | Ki | = | 107000.0 | nM | - |
| CHEMBL4448439 | — | Ki | = | 287000.0 | nM | - |
| CHEMBL4436725 | — | Ki | = | 135000.0 | nM | - |