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Assay Detail

CHEMBL4375193

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ADMET
Inhibition of N-terminal GST-tagged human EGFR (696 to end aminoacids) expressed in baculovirus infected Sf21 cells
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type Sf21
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Epidermal growth factor receptor (CHEMBL203)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton's Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological Diseases.
Caldwell RD, Qiu H, Askew BC, Bender AT, Brugger N, Camps M, Dhanabal M, Dutt V, Eichhorn T, Gardberg AS, Goutopoulos A, Grenningloh R, Head J, Healey B, Hodous BL, Huck BR, Johnson TL, Jones C, Jones RC, Mochalkin I, Morandi F, Nguyen N, Meyring M, Potnick JR, Santos DC, Schmidt R, Sherer B, Shutes A, Urbahns K, Follis AV, Wegener AA, Zimmerli SC, Liu-Bujalski L.
J Med Chem (2019) 62 : 7643 -7655
PubMed 31368705 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 7.09 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4436563 1 9.00
CHEMBL4554990 1 8.40
CHEMBL4528630 1 7.11
CHEMBL4461455 1 6.85
CHEMBL47940 1 6.75
CHEMBL4468148 1 6.26
CHEMBL4072833 EVOBRUTINIB 3.0 1 5.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4436563 IC50 = 1.0 nM 9.00
CHEMBL4554990 IC50 = 4.0 nM 8.40
CHEMBL4528630 IC50 = 78.0 nM 7.11
CHEMBL4461455 IC50 = 140.0 nM 6.85
CHEMBL47940 IC50 = 177.0 nM 6.75
CHEMBL4468148 IC50 = 550.0 nM 6.26
CHEMBL4072833 EVOBRUTINIB IC50 = 5800.0 nM 5.24