Assay Detail
Functional
CHEMBL4375365
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Antiproliferative activity against human Calu6 cells measured after 48 hrs by MTT assay
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Calu-6 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of Inhibitors of Aurora/PLK Targets as Anticancer Agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Activity | 2 | - | - |
| IC50 | 1 | 5.28 | 5.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4445812 | — | — | 1 | 5.28 |
| CHEMBL4459711 | — | — | 1 | - |
| CHEMBL4557342 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4445812 | — | IC50 | = | 5300.0 | nM | 5.28 |
| CHEMBL4459711 | — | Activity | - | — | - | |
| CHEMBL4557342 | — | Activity | - | — | - |