Assay Detail
Functional
CHEMBL4384569
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Antiproliferative activity against human HL60 cells after 72 hrs by CCK8 assay
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A Pair of Enantiomeric Bis- seco-abietane Diterpenoids from Cryptomeria fortunei.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 12 | 5.24 | 10.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL58 | MITOXANTRONE | 4.0 | 1 | 10.62 |
| CHEMBL4553108 | — | — | 1 | 4.80 |
| CHEMBL4471013 | — | — | 1 | 4.76 |
| CHEMBL4582949 | — | — | 1 | 4.68 |
| CHEMBL4474104 | — | — | 1 | 4.66 |
| CHEMBL4435892 | — | — | 1 | 4.59 |
| CHEMBL4469547 | — | — | 1 | 4.38 |
| CHEMBL4449186 | — | — | 1 | 4.34 |
| CHEMBL4594115 | — | — | 1 | 4.31 |
| CHEMBL494660 | — | — | 1 | - |
| CHEMBL4482875 | — | — | 1 | - |
| CHEMBL4469911 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL58 | MITOXANTRONE | IC50 | = | 0.024 | nM | 10.62 |
| CHEMBL4553108 | — | IC50 | = | 16000.0 | nM | 4.80 |
| CHEMBL4471013 | — | IC50 | = | 17200.0 | nM | 4.76 |
| CHEMBL4582949 | — | IC50 | = | 20800.0 | nM | 4.68 |
| CHEMBL4474104 | — | IC50 | = | 21700.0 | nM | 4.66 |
| CHEMBL4435892 | — | IC50 | = | 25700.0 | nM | 4.59 |
| CHEMBL4469547 | — | IC50 | = | 41200.0 | nM | 4.38 |
| CHEMBL4449186 | — | IC50 | = | 45500.0 | nM | 4.34 |
| CHEMBL4594115 | — | IC50 | = | 49400.0 | nM | 4.31 |
| CHEMBL494660 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4482875 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4469911 | — | IC50 | > | 100000.0 | nM | - |