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Assay Detail

CHEMBL4385022

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ADMET
Cytotoxicity against human WI38 cells assessed as reduction in cell viability after 48 hrs by MTT assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type WI-38
Confidence 1 — Organism
Curated By Autocuration

Target

WI-38 (CHEMBL614391)
Type CELL-LINE
Organism Homo sapiens

Publication

Melanogenesis-Inhibitory and Cytotoxic Activities of Triterpene Glycoside Constituents from the Bark of Albizia procera.
Zhang J, Akihisa T, Kurita M, Kikuchi T, Zhu WF, Ye F, Dong ZH, Liu WY, Feng F, Xu J.
J Nat Prod (2018) 81 : 2612 -2620
PubMed 30520635 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.39 5.66

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4451985 1 5.66
CHEMBL4561300 1 5.60
CHEMBL4581280 1 5.32
CHEMBL4483588 1 5.29
CHEMBL4448517 1 5.08

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4451985 IC50 = 2200.0 nM 5.66
CHEMBL4561300 IC50 = 2500.0 nM 5.60
CHEMBL4581280 IC50 = 4800.0 nM 5.32
CHEMBL4483588 IC50 = 5100.0 nM 5.29
CHEMBL4448517 IC50 = 8300.0 nM 5.08