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Assay Detail

CHEMBL4392265

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Binding
Inhibition of recombinant rat C-terminal His-tagged soluble form of CD73 expressed in baculovirus infected Sf9 insect cells using [2,8-3H]AMP as substrate measured after 25 mins by scintillation counting method
51
Total Activities
51
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Cell Type Sf9
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5'-nucleotidase (CHEMBL1075214)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Structure-Activity Relationship of Purine and Pyrimidine Nucleotides as Ecto-5'-Nucleotidase (CD73) Inhibitors.
Junker A, Renn C, Dobelmann C, Namasivayam V, Jain S, Losenkova K, Irjala H, Duca S, Balasubramanian R, Chakraborty S, Börgel F, Zimmermann H, Yegutkin GG, Müller CE, Jacobson KA.
J Med Chem (2019) 62 : 3677 -3695
PubMed 30895781 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 51 6.65 8.44

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4443977 1 8.44
CHEMBL4483379 1 7.86
CHEMBL3606064 1 7.83
CHEMBL4443094 1 7.73
CHEMBL4551648 1 7.52
CHEMBL4470616 1 7.07
CHEMBL4538320 1 7.06
CHEMBL4561816 1 7.05
CHEMBL4457058 1 7.05
CHEMBL4299847 1 6.95
CHEMBL1198914 1 6.79
CHEMBL583969 PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER 1 6.78
CHEMBL1198873 1 6.59
CHEMBL4440236 1 6.58
CHEMBL4462889 1 6.56
CHEMBL4474742 1 6.49
CHEMBL3606109 1 6.47
CHEMBL4441328 1 6.46
CHEMBL4574475 1 6.37
CHEMBL4436640 1 6.30
CHEMBL4543740 1 6.19
CHEMBL4587157 1 6.11
CHEMBL3220831 1 6.05
CHEMBL4472359 1 5.98
CHEMBL4530172 1 5.76
CHEMBL507060 1 5.74
CHEMBL3606055 1 5.73
CHEMBL4565565 1 5.71
CHEMBL4516688 1 5.69
CHEMBL4443859 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4443977 Ki = 3.67 nM 8.44
CHEMBL4483379 Ki = 13.9 nM 7.86
CHEMBL3606064 Ki = 14.8 nM 7.83
CHEMBL4443094 Ki = 18.8 nM 7.73
CHEMBL4551648 Ki = 30.3 nM 7.52
CHEMBL4470616 Ki = 85.1 nM 7.07
CHEMBL4538320 Ki = 86.7 nM 7.06
CHEMBL4561816 Ki = 88.6 nM 7.05
CHEMBL4457058 Ki = 88.7 nM 7.05
CHEMBL4299847 Ki = 112.0 nM 6.95
CHEMBL1198914 Ki = 162.0 nM 6.79
CHEMBL583969 PHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER Ki = 167.0 nM 6.78
CHEMBL1198873 Ki = 257.0 nM 6.59
CHEMBL4440236 Ki = 262.0 nM 6.58
CHEMBL4462889 Ki = 276.0 nM 6.56
CHEMBL4474742 Ki = 321.0 nM 6.49
CHEMBL3606109 Ki = 338.0 nM 6.47
CHEMBL4441328 Ki = 349.0 nM 6.46
CHEMBL4574475 Ki = 424.0 nM 6.37
CHEMBL4436640 Ki = 502.0 nM 6.30
CHEMBL4543740 Ki = 639.0 nM 6.19
CHEMBL4587157 Ki = 780.0 nM 6.11
CHEMBL3220831 Ki = 898.0 nM 6.05
CHEMBL4472359 Ki = 1050.0 nM 5.98
CHEMBL4530172 Ki = 1750.0 nM 5.76
CHEMBL507060 Ki = 1830.0 nM 5.74
CHEMBL3606055 Ki = 1860.0 nM 5.73
CHEMBL4565565 Ki = 1970.0 nM 5.71
CHEMBL4516688 Ki = 2030.0 nM 5.69
CHEMBL4458332 Ki > 1000.0 nM -
CHEMBL4537717 Ki > 1000.0 nM -
CHEMBL4449088 Ki > 1000.0 nM -
CHEMBL1198696 Ki > 1000.0 nM -
CHEMBL4442307 Ki > 1000.0 nM -
CHEMBL4448168 Ki > 1000.0 nM -
CHEMBL4471653 Ki > 1000.0 nM -
CHEMBL1199783 Ki > 1000.0 nM -
CHEMBL4459165 Ki > 1000.0 nM -
CHEMBL4442199 Ki > 1000.0 nM -
CHEMBL1236535 Ki > 1000.0 nM -
CHEMBL4468019 Ki > 1000.0 nM -
CHEMBL4451900 Ki > 1000.0 nM -
CHEMBL4474595 Ki > 1000.0 nM -
CHEMBL4476067 Ki > 1000.0 nM -
CHEMBL4463295 Ki > 1000.0 nM -
CHEMBL4592397 Ki > 1000.0 nM -
CHEMBL4516140 Ki > 1000.0 nM -
CHEMBL4587724 Ki > 1000.0 nM -
CHEMBL4472287 Ki > 1000.0 nM -
CHEMBL4443859 Ki > 1000.0 nM -