Assay Detail
Binding
CHEMBL4398442
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Inhibition of sulfatase (unknown origin) using [3H]DHEAS as substrate after 18 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Estrogen signaling: An emanating therapeutic target for breast cancer treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.62 | 8.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1627465 | — | — | 1 | 8.85 |
| CHEMBL1627878 | — | — | 1 | 8.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1627465 | — | IC50 | = | 1.4 | nM | 8.85 |
| CHEMBL1627878 | — | IC50 | = | 4.1 | nM | 8.39 |