Assay Detail
Binding
CHEMBL4398460
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Inhibition of adenosine receptor A1 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The chemical biology of apoptosis: Revisited after 17 years.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.11 | 6.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1269107 | — | — | 1 | 6.91 |
| CHEMBL408194 | OBATOCLAX | 3.0 | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1269107 | — | Ki | = | 122.0 | nM | 6.91 |
| CHEMBL408194 | OBATOCLAX | Ki | = | 5000.0 | nM | 5.30 |