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Assay Detail

CHEMBL4399036

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human steroid sulfatase by fluorimetric assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Steryl-sulfatase (CHEMBL3559)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Sulfamates in drug design and discovery: Pre-clinical and clinical investigations.
Zaraei SO, Abduelkarem AR, Anbar HS, Kobeissi S, Mohammad M, Ossama A, El-Gamal MI.
Eur J Med Chem (2019) 179 : 257 -271
PubMed 31255926 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 9.47 9.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL262050 1 9.47

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL262050 IC50 = 0.34 nM 9.47