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Assay Detail

CHEMBL4403370

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against Leishmania mexicana intracellular amastigotes infected in J774 macrophages assessed as reduction in parasite viability after 72 hrs
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania mexicana
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania mexicana (CHEMBL612880)
Type ORGANISM
Organism Leishmania mexicana

Publication

Multi-target drugs active against leishmaniasis: A paradigm of drug repurposing.
Braga SS.
Eur J Med Chem (2019) 183 : 111660 -111660
PubMed 31514064 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.96 7.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL561057 SQ109 2.0 1 7.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL561057 SQ109 IC50 = 11.0 nM 7.96