Assay Detail
Binding
CHEMBL4403612
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of AmpC beta-lactamase (unknown origin) by Cheng-Prusoff equation analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacteria |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
β-Lactamase Inhibitors To Restore the Efficacy of Antibiotics against Superbugs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.70 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4209255 | — | — | 1 | 10.30 |
| CHEMBL4206040 | — | — | 1 | 9.70 |
| CHEMBL4217629 | — | — | 1 | 9.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4209255 | — | Ki | = | 0.05 | nM | 10.30 |
| CHEMBL4206040 | — | Ki | = | 0.2 | nM | 9.70 |
| CHEMBL4217629 | — | Ki | = | 0.8 | nM | 9.10 |