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Assay Detail

CHEMBL4406530

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ADMET
Displacement of [3H]-methylspiperon from human D2RL expressed in HEK293 cell membranes measured after 90 mins by topcount assay
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HEK293
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

D(2) dopamine receptor (CHEMBL217)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery, Optimization, and Characterization of ML417: A Novel and Highly Selective D3 Dopamine Receptor Agonist.
Moritz AE, Free RB, Weiner WS, Akano EO, Gandhi D, Abramyan A, Keck TM, Ferrer M, Hu X, Southall N, Steiner J, Aubé J, Shi L, Frankowski KJ, Sibley DR.
J Med Chem (2020) 63 : 5526 -5567
PubMed 32342685 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 8.01 8.33
IC50 1 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL301265 PRAMIPEXOLE 4.0 1 8.33
CHEMBL2203406 1 7.68
CHEMBL1700053 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL301265 PRAMIPEXOLE Ki = 4.7 nM 8.33
CHEMBL2203406 Ki = 21.0 nM 7.68
CHEMBL1700053 IC50 > 100000.0 nM -