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Assay Detail

CHEMBL4407776

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Zika virus PRVABC59 infected in human A549 cells assessed as reduction in viral titer incubated for 48 hrs by plague assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Zika virus
Confidence 1 — Organism
Curated By Autocuration

Target

Zika virus (CHEMBL4296612)
Type ORGANISM
Organism Zika virus

Publication

Cell-active carbazole derivatives as inhibitors of the zika virus protease.
Rassias G, Zogali V, Swarbrick CMD, Ki Chan KW, Chan SA, Gwee CP, Wang S, Kaplanai E, Canko A, Kiousis D, Lescar J, Luo D, Matsoukas MT, Vasudevan SG.
Eur J Med Chem (2019) 180 : 536 -545
PubMed 31344613 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.00 6.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4437334 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4437334 EC50 = 1000.0 nM 6.00