Assay Detail
Functional
CHEMBL4410898
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Cytotoxicity against human SUDHL6 cells assessed as reduction in cell viability incubated for 4 days by celltiter glo luminescent assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SU-DHL-6 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
INCB050465 (Parsaclisib), a Novel Next-Generation Inhibitor of Phosphoinositide 3-Kinase Delta (PI3Kδ).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 7.54 | 9.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4574593 | — | — | 1 | 9.33 |
| CHEMBL4297615 | PARSACLISIB | 3.0 | 1 | 8.80 |
| CHEMBL4561896 | — | — | 1 | 8.68 |
| CHEMBL4593387 | — | — | 1 | 8.62 |
| CHEMBL4438376 | — | — | 1 | 8.51 |
| CHEMBL4458634 | — | — | 1 | 8.13 |
| CHEMBL4443149 | — | — | 1 | 7.89 |
| CHEMBL4446120 | — | — | 1 | 7.85 |
| CHEMBL2216863 | DEZAPELISIB | 2.0 | 1 | 7.75 |
| CHEMBL4444112 | — | — | 1 | 7.68 |
| CHEMBL4465303 | — | — | 1 | 7.36 |
| CHEMBL4570334 | — | — | 1 | 7.22 |
| CHEMBL4471294 | — | — | 1 | 7.14 |
| CHEMBL4513857 | — | — | 1 | 7.00 |
| CHEMBL4440146 | — | — | 1 | 6.85 |
| CHEMBL4470672 | — | — | 1 | 6.77 |
| CHEMBL4468580 | — | — | 1 | 6.08 |
| CHEMBL4576207 | — | — | 1 | 5.89 |
| CHEMBL4593849 | — | — | 1 | 5.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4574593 | — | IC50 | = | 0.47 | nM | 9.33 |
| CHEMBL4297615 | PARSACLISIB | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL4561896 | — | IC50 | = | 2.1 | nM | 8.68 |
| CHEMBL4593387 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL4438376 | — | IC50 | = | 3.1 | nM | 8.51 |
| CHEMBL4458634 | — | IC50 | = | 7.4 | nM | 8.13 |
| CHEMBL4443149 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4446120 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL2216863 | DEZAPELISIB | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4444112 | — | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL4465303 | — | IC50 | = | 44.0 | nM | 7.36 |
| CHEMBL4570334 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL4471294 | — | IC50 | = | 73.0 | nM | 7.14 |
| CHEMBL4513857 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4440146 | — | IC50 | = | 140.0 | nM | 6.85 |
| CHEMBL4470672 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL4468580 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL4576207 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL4593849 | — | IC50 | = | 1800.0 | nM | 5.75 |