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Assay Detail

CHEMBL4411348

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of tyrosinase in mouse B16 cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Tyrosinase (CHEMBL5346)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Inhibitors of Melanogenesis: An Updated Review.
Pillaiyar T, Namasivayam V, Manickam M, Jung SH.
J Med Chem (2018) 61 : 7395 -7418
PubMed 29763564 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 6.13 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL221291 1 6.52
CHEMBL4445400 1 6.10
CHEMBL43065 OXYRESVERATROL 1 5.77
CHEMBL455619 MULBERROSIDE A 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL221291 IC50 = 300.0 nM 6.52
CHEMBL4445400 IC50 = 800.0 nM 6.10
CHEMBL43065 OXYRESVERATROL IC50 = 1700.0 nM 5.77
CHEMBL455619 MULBERROSIDE A IC50 > 100000.0 nM -