Assay Detail
Binding
CHEMBL4418462
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant His-tagged human ATG7 incubated for 105 mins in presence of GST-tagged ATG3 and Flag-tagged Gabarap and measured after 2 hrs by FRET assay
230
Total Activities
228
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ubiquitin-like modifier-activating enzyme ATG7 (CHEMBL2321621) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Atg7 inhibitors and the uses thereof
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 230 | 7.35 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4467807 | — | — | 1 | 7.70 |
| CHEMBL4577562 | — | — | 1 | 7.70 |
| CHEMBL4579107 | — | — | 1 | 7.70 |
| CHEMBL4535927 | — | — | 1 | 7.70 |
| CHEMBL4521754 | — | — | 1 | 7.70 |
| CHEMBL4434940 | — | — | 1 | 7.70 |
| CHEMBL4449861 | — | — | 1 | 7.70 |
| CHEMBL4527646 | — | — | 1 | 7.70 |
| CHEMBL4546984 | — | — | 1 | 7.70 |
| CHEMBL4550475 | — | — | 1 | 7.70 |
| CHEMBL4557103 | — | — | 1 | 7.70 |
| CHEMBL4576658 | — | — | 1 | 7.70 |
| CHEMBL4471077 | — | — | 1 | 7.70 |
| CHEMBL4449596 | — | — | 1 | 7.70 |
| CHEMBL4483085 | — | — | 1 | 7.70 |
| CHEMBL4466430 | — | — | 1 | 7.70 |
| CHEMBL4557469 | — | — | 1 | 7.70 |
| CHEMBL4452757 | — | — | 1 | 7.70 |
| CHEMBL4518269 | — | — | 1 | 7.70 |
| CHEMBL4518410 | — | — | 1 | 7.70 |
| CHEMBL4537063 | — | — | 1 | 7.70 |
| CHEMBL4473356 | — | — | 1 | 7.70 |
| CHEMBL4526319 | — | — | 1 | 7.70 |
| CHEMBL4456716 | — | — | 1 | 7.70 |
| CHEMBL4543610 | — | — | 1 | 7.70 |
| CHEMBL4447381 | — | — | 1 | 7.70 |
| CHEMBL4558671 | — | — | 1 | 7.70 |
| CHEMBL4464322 | — | — | 1 | 7.70 |
| CHEMBL4457043 | — | — | 1 | 7.70 |
| CHEMBL4454053 | — | — | 1 | 7.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4467807 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4589617 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4539628 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4557103 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4542158 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4576658 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4439106 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4471077 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4575995 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4476516 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4451742 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4483085 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4558671 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4436997 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4473245 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4526319 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4456716 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4453903 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4543610 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4475447 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4447381 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4548069 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4466430 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4589191 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4454053 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4434940 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4476015 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4589701 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4469589 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4551253 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4577562 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4579107 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4451885 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4535927 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4529186 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4468221 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4521754 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4469119 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4449596 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4449861 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4444895 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4532634 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4517771 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4574054 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4455332 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4527646 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4546984 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4550475 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4545152 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4551395 | — | IC50 | = | 20.0 | nM | 7.70 |