Assay Detail
Functional
CHEMBL4419274
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human NCI-H226 cells incubated for 3 days
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H226 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Methods and compositions for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 4.27 | 4.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2030270 | — | — | 1 | 4.89 |
| CHEMBL4442569 | — | — | 1 | 4.72 |
| CHEMBL4576938 | — | — | 1 | 4.36 |
| CHEMBL4515226 | — | — | 1 | 4.26 |
| CHEMBL4464276 | — | — | 1 | 4.22 |
| CHEMBL4529653 | — | — | 1 | 4.22 |
| CHEMBL4552833 | — | — | 1 | 4.22 |
| CHEMBL4577791 | — | — | 1 | 4.19 |
| CHEMBL4552253 | — | — | 1 | 4.19 |
| CHEMBL4451129 | — | — | 1 | 4.16 |
| CHEMBL4437164 | — | — | 1 | 4.16 |
| CHEMBL4439996 | — | — | 1 | 4.12 |
| CHEMBL4463075 | — | — | 1 | 4.02 |
| CHEMBL4472256 | — | — | 1 | 4.02 |
| CHEMBL4446354 | — | — | 1 | - |
| CHEMBL4528582 | — | — | 1 | - |
| CHEMBL4542845 | — | — | 1 | - |
| CHEMBL4542842 | — | — | 1 | - |
| CHEMBL4435105 | — | — | 1 | - |
| CHEMBL4519349 | — | — | 1 | - |
| CHEMBL4280751 | — | — | 1 | - |
| CHEMBL4280394 | — | — | 1 | - |
| CHEMBL4279325 | — | — | 1 | - |
| CHEMBL4293794 | — | — | 1 | - |
| CHEMBL4283567 | — | — | 1 | - |
| CHEMBL4474905 | — | — | 1 | - |
| CHEMBL4287230 | — | — | 1 | - |
| CHEMBL4451466 | — | — | 1 | - |
| CHEMBL4282142 | — | — | 1 | - |
| CHEMBL4473695 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2030270 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL4442569 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL4576938 | — | IC50 | = | 44000.0 | nM | 4.36 |
| CHEMBL4515226 | — | IC50 | = | 55000.0 | nM | 4.26 |
| CHEMBL4464276 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL4529653 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL4552833 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL4577791 | — | IC50 | = | 65000.0 | nM | 4.19 |
| CHEMBL4552253 | — | IC50 | = | 65000.0 | nM | 4.19 |
| CHEMBL4451129 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL4437164 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL4439996 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL4463075 | — | IC50 | = | 95000.0 | nM | 4.02 |
| CHEMBL4472256 | — | IC50 | = | 95000.0 | nM | 4.02 |
| CHEMBL4561494 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4454755 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4288751 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4285086 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1422005 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4446354 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4528582 | — | IC50 | >= | 52000.0 | nM | - |
| CHEMBL4542845 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4542842 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4435105 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4519349 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4280751 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4280394 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4279325 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4293794 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4283567 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4474905 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4287230 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4451466 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4282142 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4473695 | — | IC50 | > | 100000.0 | nM | - |