Assay Detail
Functional
CHEMBL4419287
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Growth inhibition of human A549 cells incubated for 3 days
31
Total Activities
31
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A549 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Methods and compositions for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 31 | 4.46 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4285086 | — | — | 1 | 5.70 |
| CHEMBL4288751 | — | — | 1 | 5.52 |
| CHEMBL1422005 | — | — | 1 | 4.82 |
| CHEMBL4464276 | — | — | 1 | 4.60 |
| CHEMBL4442569 | — | — | 1 | 4.57 |
| CHEMBL4552253 | — | — | 1 | 4.57 |
| CHEMBL4515226 | — | — | 1 | 4.52 |
| CHEMBL4577791 | — | — | 1 | 4.42 |
| CHEMBL4528582 | — | — | 1 | 4.38 |
| CHEMBL4529653 | — | — | 1 | 4.35 |
| CHEMBL4472256 | — | — | 1 | 4.30 |
| CHEMBL4519349 | — | — | 1 | 4.29 |
| CHEMBL4451129 | — | — | 1 | 4.26 |
| CHEMBL4439996 | — | — | 1 | 4.22 |
| CHEMBL4552833 | — | — | 1 | 4.14 |
| CHEMBL4451466 | — | — | 1 | 4.12 |
| CHEMBL4542842 | — | — | 1 | 4.05 |
| CHEMBL4437164 | — | — | 1 | 4.00 |
| CHEMBL4435105 | — | — | 1 | 4.00 |
| CHEMBL4463075 | — | — | 1 | - |
| CHEMBL4280751 | — | — | 1 | - |
| CHEMBL4454755 | — | — | 1 | - |
| CHEMBL4561494 | — | — | 1 | - |
| CHEMBL4280394 | — | — | 1 | - |
| CHEMBL4279325 | — | — | 1 | - |
| CHEMBL4293794 | — | — | 1 | - |
| CHEMBL4474905 | — | — | 1 | - |
| CHEMBL4282142 | — | — | 1 | - |
| CHEMBL4283567 | — | — | 1 | - |
| CHEMBL4473695 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4285086 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL4288751 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1422005 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL4464276 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL4442569 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL4552253 | — | IC50 | = | 27000.0 | nM | 4.57 |
| CHEMBL4515226 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL4577791 | — | IC50 | = | 38000.0 | nM | 4.42 |
| CHEMBL4528582 | — | IC50 | = | 42000.0 | nM | 4.38 |
| CHEMBL4529653 | — | IC50 | = | 45000.0 | nM | 4.35 |
| CHEMBL4472256 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL4519349 | — | IC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL4451129 | — | IC50 | = | 55000.0 | nM | 4.26 |
| CHEMBL4439996 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL4552833 | — | IC50 | = | 72000.0 | nM | 4.14 |
| CHEMBL4451466 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL4542842 | — | IC50 | = | 90000.0 | nM | 4.05 |
| CHEMBL4437164 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL4435105 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL4463075 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4280751 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4454755 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4561494 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4280394 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4279325 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4293794 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4474905 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4282142 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4283567 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4473695 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL4287230 | — | IC50 | > | 100000.0 | nM | - |