Assay Detail
Binding
CHEMBL4419837
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Inhibition of FLAG-tagged DGKa (unknown origin) using lipids and [gamma-32P]-ATP incubated for 15 mins by scintillation counting method
4
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Compositions and methods for treating cancer
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 2 | - | - |
| IC50 | 2 | 4.88 | 5.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL267777 | RITANSERIN | 2.0 | 2 | 5.05 |
| CHEMBL259388 | — | — | 2 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL267777 | RITANSERIN | IC50 | = | 9000.0 | nM | 5.05 |
| CHEMBL259388 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL267777 | RITANSERIN | Inhibition | - | % | - | |
| CHEMBL259388 | — | Inhibition | - | % | - |