Assay Detail
Binding
CHEMBL4420299
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Binding affinity to TFPI (unknown origin) incubated for 1.5 hrs using tracer peptide JBT2271 by competition ELISA
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Tfpi inhibitors and methods of use
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.54 | 8.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4545581 | — | — | 1 | 8.54 |
| CHEMBL4473203 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4545581 | — | IC50 | = | 2.9 | nM | 8.54 |
| CHEMBL4473203 | — | IC50 | >= | 4.8 | nM | - |