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Assay Detail

CHEMBL4427461

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antitubercular activity against oxygen-deprived Mycobacterium tuberculosis H37Rv assessed as bacterial growth inhibition incubated for 5 days under aerobic conditions by LOR assay
4
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mycobacterium tuberculosis
Confidence 1 — Organism
Curated By Autocuration

Target

Mycobacterium tuberculosis (CHEMBL360)
Type ORGANISM
Organism Mycobacterium tuberculosis

Publication

Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising Class of Antimycobacterial Agents.
Hampannavar GA, Karpoormath R, Palkar MB, Shaikh MS, Chandrasekaran B.
ACS Med Chem Lett (2016) 7 : 686 -691
PubMed 27437078 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
MIC 2 - -
IC50 2 6.92 7.01

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4455126 2 7.01
CHEMBL4534306 2 6.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4455126 IC50 = 97.0 nM 7.01
CHEMBL4534306 IC50 = 150.0 nM 6.82
CHEMBL4455126 MIC = 280.0 nM -
CHEMBL4534306 MIC = 500.0 nM -