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Assay Detail

CHEMBL4428368

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Competitive inhibition of Leishmania amazonensis arginase assessed as inhibition constant for enzyme-inhibitor complex using L-arginine as substrate incubated for 15 mins by Dixon plot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Leishmania amazonensis
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Arginase (CHEMBL3108635)
Type SINGLE PROTEIN
Organism Leishmania amazonensis

Publication

Verbascoside Inhibits Promastigote Growth and Arginase Activity of Leishmania amazonensis.
Maquiaveli CC, Lucon-Júnior JF, Brogi S, Campiani G, Gemma S, Vieira PC, Silva ER.
J Nat Prod (2016) 79 : 1459 -1463
PubMed 27096224 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.16 6.16

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL444478 ACETOSIDE 2.0 1 6.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL444478 ACETOSIDE Ki = 700.0 nM 6.16