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Assay Detail

CHEMBL4431480

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of SKF-86002 binding to human inactive p38alpha after 60 mins by fluorescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Mitogen-activated protein kinase 14 (CHEMBL260)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Medchemcomm (2016) 7 : 1421 -1428
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 10.00 10.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL103667 DORAMAPIMOD 2.0 1 10.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL103667 DORAMAPIMOD Kd = 0.1 nM 10.00