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Assay Detail

CHEMBL4431573

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Binding
Inhibition of Dengue virus ribose 2'-O methyltransferase using RNA substrate after 20 mins in presence of [methyl-3H]-AdoMet by microbeta counting analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Dengue virus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Nonstructural protein 5 (CHEMBL4295629)
Type SINGLE PROTEIN
Organism Dengue virus

Publication

The Medicinal Chemistry of Dengue Virus.
Behnam MA, Nitsche C, Boldescu V, Klein CD.
J Med Chem (2016) 59 : 5622 -5649
PubMed 26771861 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.85 7.39

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1214186 SINEFUNGIN 2.0 1 7.39
CHEMBL418052 S-ADENOSYLHOMOCYSTEINE 1 6.31

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1214186 SINEFUNGIN IC50 = 41.0 nM 7.39
CHEMBL418052 S-ADENOSYLHOMOCYSTEINE IC50 = 490.0 nM 6.31