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Assay Detail

CHEMBL4431707

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Functional
Cytotoxicity against human HeLaS3 cells assessed as decrease in cell viability after 72 to 96 hrs by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HeLa S3
Confidence 1 — Organism
Curated By Autocuration

Target

HeLa S3 (CHEMBL4296436)
Type CELL-LINE
Organism Homo sapiens

Publication

Dehydroleucodine, a Sesquiterpene Lactone from Gynoxys verrucosa, Demonstrates Cytotoxic Activity against Human Leukemia Cells.
Ordóñez PE, Sharma KK, Bystrom LM, Alas MA, Enriquez RG, Malagón O, Jones DE, Guzman ML, Compadre CM.
J Nat Prod (2016) 79 : 691 -696
PubMed 27057812 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL441260 DEHYDROLEUCODIN 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL441260 DEHYDROLEUCODIN IC50 = 10000.0 nM 5.00