Assay Detail
Binding
CHEMBL4482513
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to AKT1 (unknown origin) by surface plasmon resonance assay
22
Total Activities
22
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
RAC-alpha serine/threonine-protein kinase (CHEMBL4282) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Inhibitors of grb2-associated binding protein 1 (gab1) and methods of treating cancer using the same
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 17 | 5.34 | 5.51 |
| Ki | 5 | 5.25 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL595583 | — | — | 1 | 5.62 |
| CHEMBL23552 | — | — | 1 | 5.51 |
| CHEMBL1685055 | — | — | 1 | 5.37 |
| CHEMBL4577370 | — | — | 1 | 5.34 |
| CHEMBL1685066 | — | — | 1 | 5.30 |
| CHEMBL1681823 | — | — | 1 | 5.30 |
| CHEMBL1685058 | — | — | 1 | 5.22 |
| CHEMBL3912759 | — | — | 1 | 5.20 |
| CHEMBL1685056 | — | — | 1 | 4.72 |
| CHEMBL4564787 | — | — | 1 | - |
| CHEMBL595786 | — | — | 1 | - |
| CHEMBL4539727 | — | — | 1 | - |
| CHEMBL4536878 | — | — | 1 | - |
| CHEMBL4557539 | — | — | 1 | - |
| CHEMBL4591779 | — | — | 1 | - |
| CHEMBL4530453 | — | — | 1 | - |
| CHEMBL4538899 | — | — | 1 | - |
| CHEMBL4563636 | — | — | 1 | - |
| CHEMBL4590344 | — | — | 1 | - |
| CHEMBL1572640 | — | — | 1 | - |
| CHEMBL4576057 | — | — | 1 | - |
| CHEMBL4533777 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL595583 | — | Ki | = | 2400.0 | nM | 5.62 |
| CHEMBL23552 | — | Kd | = | 3080.0 | nM | 5.51 |
| CHEMBL1685055 | — | Ki | = | 4300.0 | nM | 5.37 |
| CHEMBL4577370 | — | Kd | = | 4580.0 | nM | 5.34 |
| CHEMBL1685066 | — | Kd | = | 5040.0 | nM | 5.30 |
| CHEMBL1681823 | — | Ki | = | 5000.0 | nM | 5.30 |
| CHEMBL1685058 | — | Ki | = | 6000.0 | nM | 5.22 |
| CHEMBL3912759 | — | Kd | = | 6270.0 | nM | 5.20 |
| CHEMBL1685056 | — | Ki | = | 18900.0 | nM | 4.72 |
| CHEMBL4564787 | — | Kd | - | — | - | |
| CHEMBL595786 | — | Kd | - | — | - | |
| CHEMBL4539727 | — | Kd | - | — | - | |
| CHEMBL4536878 | — | Kd | - | — | - | |
| CHEMBL4557539 | — | Kd | - | — | - | |
| CHEMBL4591779 | — | Kd | - | — | - | |
| CHEMBL4530453 | — | Kd | - | — | - | |
| CHEMBL4538899 | — | Kd | - | — | - | |
| CHEMBL4563636 | — | Kd | - | — | - | |
| CHEMBL4590344 | — | Kd | - | — | - | |
| CHEMBL1572640 | — | Kd | - | — | - | |
| CHEMBL4576057 | — | Kd | - | — | - | |
| CHEMBL4533777 | — | Kd | - | — | - |