Assay Detail
Functional
CHEMBL4613061
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Growth inhibition of human Pfeiffer cells incubated for 7 days by WST8 assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Pfeiffer |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
EEDi-5285: An Exceptionally Potent, Efficacious, and Orally Active Small-Molecule Inhibitor of Embryonic Ectoderm Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 10.27 | 10.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4649099 | — | — | 1 | 10.70 |
| CHEMBL4637520 | — | — | 1 | 10.70 |
| CHEMBL4637096 | — | — | 1 | 10.70 |
| CHEMBL4645324 | — | — | 1 | 10.70 |
| CHEMBL4645310 | — | — | 1 | 10.52 |
| CHEMBL4638412 | — | — | 1 | 10.52 |
| CHEMBL4644746 | — | — | 1 | 10.30 |
| CHEMBL4635558 | — | — | 1 | 10.15 |
| CHEMBL4633469 | — | — | 1 | 10.10 |
| CHEMBL4643880 | — | — | 1 | 9.92 |
| CHEMBL4642335 | — | — | 1 | 9.57 |
| CHEMBL4640556 | — | — | 1 | 9.30 |
| CHEMBL4640949 | — | — | 1 | - |
| CHEMBL4647900 | — | — | 1 | - |
| CHEMBL4642454 | — | — | 1 | - |
| CHEMBL4649861 | — | — | 1 | - |
| CHEMBL4634939 | — | — | 1 | - |
| CHEMBL4639197 | — | — | 1 | - |
| CHEMBL4634654 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4649099 | — | IC50 | = | 0.02 | nM | 10.70 |
| CHEMBL4637520 | — | IC50 | = | 0.02 | nM | 10.70 |
| CHEMBL4637096 | — | IC50 | = | 0.02 | nM | 10.70 |
| CHEMBL4645324 | — | IC50 | = | 0.02 | nM | 10.70 |
| CHEMBL4645310 | — | IC50 | = | 0.03 | nM | 10.52 |
| CHEMBL4638412 | — | IC50 | = | 0.03 | nM | 10.52 |
| CHEMBL4644746 | — | IC50 | = | 0.05 | nM | 10.30 |
| CHEMBL4635558 | — | IC50 | = | 0.07 | nM | 10.15 |
| CHEMBL4633469 | — | IC50 | = | 0.08 | nM | 10.10 |
| CHEMBL4643880 | — | IC50 | = | 0.12 | nM | 9.92 |
| CHEMBL4642335 | — | IC50 | = | 0.27 | nM | 9.57 |
| CHEMBL4640556 | — | IC50 | = | 0.5 | nM | 9.30 |
| CHEMBL4640949 | — | IC50 | - | — | - | |
| CHEMBL4647900 | — | IC50 | - | — | - | |
| CHEMBL4642454 | — | IC50 | - | — | - | |
| CHEMBL4649861 | — | IC50 | - | — | - | |
| CHEMBL4634939 | — | IC50 | - | — | - | |
| CHEMBL4639197 | — | IC50 | - | — | - | |
| CHEMBL4634654 | — | IC50 | - | — | - |