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Assay Detail

CHEMBL4627508

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Binding
Agonist activity at ERalpha (unknown origin) expressed in human HeLa cells assessed as transcriptional activation measured after 24 hrs by luciferase reporter gene assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type HeLa
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Estrogen receptor (CHEMBL206)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Bisphenol AF: Halogen bonding effect is a major driving force for the dual ERα-agonist and ERβ-antagonist activities.
Liu X, Suyama K, Shiki J, Torikai K, Nose T, Shimohigashi M, Shimohigashi Y.
Bioorg Med Chem (2020) 28 : 115274 -115274
PubMed 31879182 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 7 7.63 9.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL135 ESTRADIOL 4.0 1 9.68
CHEMBL4642117 1 7.84
CHEMBL1900054 1 7.70
CHEMBL196585 1 7.51
CHEMBL4646249 1 6.96
CHEMBL418971 BISPHENOL A 1 6.10
CHEMBL2392656 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL135 ESTRADIOL EC50 = 0.21 nM 9.68
CHEMBL4642117 EC50 = 14.5 nM 7.84
CHEMBL1900054 EC50 = 20.0 nM 7.70
CHEMBL196585 EC50 = 30.7 nM 7.51
CHEMBL4646249 EC50 = 109.0 nM 6.96
CHEMBL418971 BISPHENOL A EC50 = 797.0 nM 6.10
CHEMBL2392656 EC50 > 10000.0 nM -