Assay Detail
Binding
CHEMBL4667669
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Inhibition of MALT1 (unknown origin) by Glosensor reporter gene assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mucosa-associated lymphoid tissue lymphoma translocation protein 1 (CHEMBL3632452) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Quinoline and thiazolopyridine allosteric inhibitors of MALT1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 28 | 7.18 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4784740 | — | — | 1 | 8.70 |
| CHEMBL4748253 | — | — | 1 | 8.22 |
| CHEMBL4741853 | — | — | 1 | 8.22 |
| CHEMBL4779581 | — | — | 1 | 8.15 |
| CHEMBL4762086 | — | — | 1 | 8.15 |
| CHEMBL4740000 | — | — | 1 | 7.89 |
| CHEMBL4791759 | — | — | 1 | 7.75 |
| CHEMBL4749826 | — | — | 1 | 7.57 |
| CHEMBL4751498 | — | — | 1 | 7.55 |
| CHEMBL4749854 | — | — | 1 | 7.52 |
| CHEMBL4790415 | — | — | 1 | 7.48 |
| CHEMBL4789469 | — | — | 1 | 7.46 |
| CHEMBL4784899 | — | — | 1 | 7.44 |
| CHEMBL4794268 | — | — | 1 | 7.34 |
| CHEMBL4763765 | — | — | 1 | 7.26 |
| CHEMBL4788571 | — | — | 1 | 7.16 |
| CHEMBL4742156 | — | — | 1 | 7.11 |
| CHEMBL4740768 | — | — | 1 | 7.04 |
| CHEMBL4759864 | — | — | 1 | 6.80 |
| CHEMBL4755479 | — | — | 1 | 6.78 |
| CHEMBL4782908 | — | — | 1 | 6.62 |
| CHEMBL4784606 | — | — | 1 | 6.37 |
| CHEMBL4760252 | — | — | 1 | 6.35 |
| CHEMBL4783451 | — | — | 1 | 5.70 |
| CHEMBL4799622 | — | — | 1 | 5.22 |
| CHEMBL4777911 | — | — | 1 | 4.71 |
| CHEMBL4780316 | — | — | 1 | - |
| CHEMBL4751202 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4784740 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL4748253 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL4741853 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL4779581 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4762086 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4740000 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4791759 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4749826 | — | IC50 | = | 27.0 | nM | 7.57 |
| CHEMBL4751498 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL4749854 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL4790415 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL4789469 | — | IC50 | = | 35.0 | nM | 7.46 |
| CHEMBL4784899 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL4794268 | — | IC50 | = | 46.0 | nM | 7.34 |
| CHEMBL4763765 | — | IC50 | = | 55.0 | nM | 7.26 |
| CHEMBL4788571 | — | IC50 | = | 69.0 | nM | 7.16 |
| CHEMBL4742156 | — | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL4740768 | — | IC50 | = | 92.0 | nM | 7.04 |
| CHEMBL4759864 | — | IC50 | = | 160.0 | nM | 6.80 |
| CHEMBL4755479 | — | IC50 | = | 165.0 | nM | 6.78 |
| CHEMBL4782908 | — | IC50 | = | 237.0 | nM | 6.62 |
| CHEMBL4784606 | — | IC50 | = | 432.0 | nM | 6.37 |
| CHEMBL4760252 | — | IC50 | = | 451.0 | nM | 6.35 |
| CHEMBL4783451 | — | IC50 | = | 1980.0 | nM | 5.70 |
| CHEMBL4799622 | — | IC50 | = | 6020.0 | nM | 5.22 |
| CHEMBL4777911 | — | IC50 | = | 19300.0 | nM | 4.71 |
| CHEMBL4780316 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL4751202 | — | IC50 | > | 20000.0 | nM | - |