Assay Detail
Binding
CHEMBL4672964
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Inhibition of Kca3.1 in human erythrocytes
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Intermediate conductance calcium-activated potassium channel protein 4 (CHEMBL4305) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Novel Potassium Channel Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 7.62 | 8.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4744833 | — | — | 1 | 8.09 |
| CHEMBL4749039 | — | — | 1 | 8.07 |
| CHEMBL4791725 | — | — | 1 | 8.06 |
| CHEMBL4788143 | — | — | 1 | 7.85 |
| CHEMBL4756080 | — | — | 1 | 7.75 |
| CHEMBL4764429 | — | — | 1 | 7.62 |
| CHEMBL4745327 | — | — | 1 | 7.33 |
| CHEMBL4743839 | — | — | 1 | 7.28 |
| CHEMBL4780941 | — | — | 1 | 7.12 |
| CHEMBL4785936 | — | — | 1 | 7.04 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4744833 | — | IC50 | = | 8.1 | nM | 8.09 |
| CHEMBL4749039 | — | IC50 | = | 8.6 | nM | 8.07 |
| CHEMBL4791725 | — | IC50 | = | 8.7 | nM | 8.06 |
| CHEMBL4788143 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL4756080 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4764429 | — | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL4745327 | — | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL4743839 | — | IC50 | = | 52.0 | nM | 7.28 |
| CHEMBL4780941 | — | IC50 | = | 75.0 | nM | 7.12 |
| CHEMBL4785936 | — | IC50 | = | 92.0 | nM | 7.04 |