Assay Detail
Functional
CHEMBL4675514
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antimicrobial activity against nano-luciferase-expressing Cryptosporidium parvum infected in human HCT8 cells incubated for 72 hrs by luciferase reporter gene assay
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cryptosporidium parvum |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Development of 5-Aminopyrazole-4-carboxamide-based Bumped-Kinase Inhibitors for Cryptosporidiosis Therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 27 | 6.20 | 6.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4787093 | — | — | 1 | 6.68 |
| CHEMBL4742781 | — | — | 1 | 6.60 |
| CHEMBL4791496 | — | — | 1 | 6.46 |
| CHEMBL4787718 | — | — | 1 | 6.43 |
| CHEMBL4751724 | — | — | 1 | 6.39 |
| CHEMBL4764836 | — | — | 1 | 6.38 |
| CHEMBL4796309 | — | — | 1 | 6.37 |
| CHEMBL4756756 | — | — | 1 | 6.36 |
| CHEMBL4751897 | — | — | 1 | 6.35 |
| CHEMBL4750746 | — | — | 1 | 6.31 |
| CHEMBL4743192 | — | — | 1 | 6.29 |
| CHEMBL4759936 | — | — | 1 | 6.28 |
| CHEMBL4756763 | — | — | 1 | 6.22 |
| CHEMBL4744995 | — | — | 1 | 6.19 |
| CHEMBL4750862 | — | — | 1 | 6.18 |
| CHEMBL3769570 | — | — | 1 | 6.15 |
| CHEMBL4800671 | — | — | 1 | 6.15 |
| CHEMBL4753185 | — | — | 1 | 6.15 |
| CHEMBL4749451 | — | — | 1 | 6.14 |
| CHEMBL4762379 | — | — | 1 | 6.13 |
| CHEMBL4753941 | — | — | 1 | 6.06 |
| CHEMBL3770980 | — | — | 1 | 6.05 |
| CHEMBL4740515 | — | — | 1 | 5.99 |
| CHEMBL4756120 | — | — | 1 | 5.91 |
| CHEMBL4777462 | — | — | 1 | 5.88 |
| CHEMBL3770743 | — | — | 1 | 5.74 |
| CHEMBL4750009 | — | — | 1 | 5.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4787093 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL4742781 | — | EC50 | = | 250.0 | nM | 6.60 |
| CHEMBL4791496 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL4787718 | — | EC50 | = | 370.0 | nM | 6.43 |
| CHEMBL4751724 | — | EC50 | = | 410.0 | nM | 6.39 |
| CHEMBL4764836 | — | EC50 | = | 420.0 | nM | 6.38 |
| CHEMBL4796309 | — | EC50 | = | 430.0 | nM | 6.37 |
| CHEMBL4756756 | — | EC50 | = | 440.0 | nM | 6.36 |
| CHEMBL4751897 | — | EC50 | = | 450.0 | nM | 6.35 |
| CHEMBL4750746 | — | EC50 | = | 490.0 | nM | 6.31 |
| CHEMBL4743192 | — | EC50 | = | 510.0 | nM | 6.29 |
| CHEMBL4759936 | — | EC50 | = | 530.0 | nM | 6.28 |
| CHEMBL4756763 | — | EC50 | = | 600.0 | nM | 6.22 |
| CHEMBL4744995 | — | EC50 | = | 650.0 | nM | 6.19 |
| CHEMBL4750862 | — | EC50 | = | 660.0 | nM | 6.18 |
| CHEMBL3769570 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL4800671 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL4753185 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL4749451 | — | EC50 | = | 730.0 | nM | 6.14 |
| CHEMBL4762379 | — | EC50 | = | 740.0 | nM | 6.13 |
| CHEMBL4753941 | — | EC50 | = | 880.0 | nM | 6.06 |
| CHEMBL3770980 | — | EC50 | = | 890.0 | nM | 6.05 |
| CHEMBL4740515 | — | EC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL4756120 | — | EC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL4777462 | — | EC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL3770743 | — | EC50 | = | 1820.0 | nM | 5.74 |
| CHEMBL4750009 | — | EC50 | = | 3300.0 | nM | 5.48 |