Assay Detail
Binding
CHEMBL4676746
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Inhibition of bovine adrenal medulla DBH incubated for 25 mins
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Pyridine alkaloids with activity in the central nervous system.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.36 | 7.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4764135 | — | — | 1 | 7.41 |
| CHEMBL24510 | FUSARIC ACID | — | 1 | 7.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4764135 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL24510 | FUSARIC ACID | IC50 | = | 50.0 | nM | 7.30 |