Assay Detail
Binding
CHEMBL4683693
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of alpha-glucosidase (unknown origin) using sucrose as substrate incubated for 30 mins
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of novel pyrido-pyrrolidine hybrid compounds as alpha-glucosidase inhibitors and alternative agent for control of type 1 diabetes.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.10 | 5.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL454551 | L-RADICAMINE A | — | 1 | 5.17 |
| CHEMBL4783560 | — | — | 1 | 5.03 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL454551 | L-RADICAMINE A | IC50 | = | 6700.0 | nM | 5.17 |
| CHEMBL4783560 | — | IC50 | = | 9300.0 | nM | 5.03 |