Assay Detail
Binding
CHEMBL4687295
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of mouse BTK expressed in baculovirus infected Sf21 cells incubated for 1 hr by Western blot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | Sf21 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Progress toward a Glycoprotein VI Modulator for the Treatment of Thrombosis.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.60 | 5.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL228043 | — | — | 1 | 5.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL228043 | — | IC50 | = | 2500.0 | nM | 5.60 |