Assay Detail
Binding
CHEMBL4687754
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of MDM2 (unknown origin) by cell-based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Opportunities for Tapping into Three-Dimensional Chemical Space through a Quaternary Carbon.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.00 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2381408 | SAR-405838 | 1.0 | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2381408 | SAR-405838 | IC50 | = | 100.0 | nM | 7.00 |