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Assay Detail

CHEMBL4701430

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Functional
Antiproliferative activity against human MOLM-13 cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MOLM-13
Confidence 1 — Organism
Curated By Autocuration

Target

MOLM-13 (CHEMBL3706572)
Type CELL-LINE
Organism Homo sapiens

Publication

Recent Developments in the Biology and Medicinal Chemistry of CDK9 Inhibitors: An Update.
Wu T,Qin Z,Tian Y,Wang J,Xu C,Li Z,Bian J
J Med Chem (2020) 63 : 13228 -13257
PubMed 32866383 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.54 7.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4756595 ENITOCICLIB 1.0 1 7.54

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4756595 ENITOCICLIB IC50 = 29.0 nM 7.54