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Assay Detail

CHEMBL4713445

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Binding
Binding affinity to 5HT1A receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 1A (CHEMBL214)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-Activity Relationship and Biological Investigation of SR18292 (16), a Suppressor of Glucagon-Induced Glucose Production.
Lin H,Sharabi K,Lin L,Ruiz C,Zhu D,Cameron MD,Novick SJ,Griffin PR,Puigserver P,Kamenecka TM
J Med Chem (2021) 64 : 980 -990
PubMed 33434430 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.68 5.68

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4789047 1 5.68

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4789047 Ki = 2100.0 nM 5.68