Assay Detail
Binding
CHEMBL4714150
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of DPP9 (unknown origin) using AMC substrate by fluorometric assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification of BR102910 as a selective fibroblast activation protein (FAP) inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.90 | 4.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3233842 | — | — | 1 | 4.90 |
| CHEMBL4747683 | — | — | 1 | - |
| CHEMBL2333026 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3233842 | — | IC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL4747683 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL2333026 | — | IC50 | > | 100000.0 | nM | - |