Assay Detail
ADMET
CHEMBL4716833
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Antiproliferative activity against wild type mouse BaF3 cells assessed as reduction in cell growth incubated for 2 to 3 days by Bright-Glo luciferase assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | BaF3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Design and synthesis of novel selective anaplastic lymphoma kinase inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 5.41 | 5.69 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4795530 | — | — | 1 | 5.69 |
| CHEMBL4779222 | — | — | 1 | 5.65 |
| CHEMBL2403108 | CERITINIB | 4.0 | 1 | 5.61 |
| CHEMBL3651854 | — | — | 1 | 5.60 |
| CHEMBL4739938 | — | — | 1 | 5.58 |
| CHEMBL4749543 | — | — | 1 | 5.49 |
| CHEMBL4762256 | — | — | 1 | 5.47 |
| CHEMBL3734798 | — | — | 1 | 5.46 |
| CHEMBL4762929 | — | — | 1 | 5.41 |
| CHEMBL4755518 | — | — | 1 | 5.35 |
| CHEMBL4787280 | — | — | 1 | 5.31 |
| CHEMBL4798141 | — | — | 1 | 5.29 |
| CHEMBL4780490 | — | — | 1 | 5.27 |
| CHEMBL4762861 | — | — | 1 | 5.26 |
| CHEMBL4756013 | — | — | 1 | 5.24 |
| CHEMBL4791252 | — | — | 1 | 5.21 |
| CHEMBL4747015 | — | — | 1 | 5.14 |
| CHEMBL3651885 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4795530 | — | IC50 | = | 2033.0 | nM | 5.69 |
| CHEMBL4779222 | — | IC50 | = | 2216.0 | nM | 5.65 |
| CHEMBL2403108 | CERITINIB | IC50 | = | 2477.0 | nM | 5.61 |
| CHEMBL3651854 | — | IC50 | = | 2507.0 | nM | 5.60 |
| CHEMBL4739938 | — | IC50 | = | 2599.0 | nM | 5.58 |
| CHEMBL4749543 | — | IC50 | = | 3240.0 | nM | 5.49 |
| CHEMBL4762256 | — | IC50 | = | 3422.0 | nM | 5.47 |
| CHEMBL3734798 | — | IC50 | = | 3479.0 | nM | 5.46 |
| CHEMBL4762929 | — | IC50 | = | 3940.0 | nM | 5.41 |
| CHEMBL4755518 | — | IC50 | = | 4503.0 | nM | 5.35 |
| CHEMBL4787280 | — | IC50 | = | 4912.0 | nM | 5.31 |
| CHEMBL4798141 | — | IC50 | = | 5120.0 | nM | 5.29 |
| CHEMBL4780490 | — | IC50 | = | 5411.0 | nM | 5.27 |
| CHEMBL4762861 | — | IC50 | = | 5540.0 | nM | 5.26 |
| CHEMBL4756013 | — | IC50 | = | 5731.0 | nM | 5.24 |
| CHEMBL4791252 | — | IC50 | = | 6220.0 | nM | 5.21 |
| CHEMBL4747015 | — | IC50 | = | 7230.0 | nM | 5.14 |
| CHEMBL3651885 | — | IC50 | > | 10000.0 | nM | - |