Assay Detail
Functional
CHEMBL4723153
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Antiviral activity against HCoV-NL63 infected in Rhesus macaque LLC-MK2 cells incubated for 72 hrs by RT-PCR method
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human coronavirus NL63 |
| Cell Type | LLC-MK2 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Chinese Therapeutic Strategy for Fighting COVID-19 and Potential Small-Molecule Inhibitors against Severe Acute Respiratory Syndrome Coronavirus 2 (SARS-CoV-2).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 7 | 6.08 | 6.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL866 | MYCOPHENOLIC ACID | 4.0 | 1 | 6.75 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | 4.0 | 1 | 6.64 |
| CHEMBL400092 | LYCORINE | — | 1 | 6.33 |
| CHEMBL50588 | EMETINE | 4.0 | 1 | 5.84 |
| CHEMBL5314365 | MONENSIN SODIUM | 4.0 | 1 | 5.81 |
| CHEMBL1242 | PHENAZOPYRIDINE | 4.0 | 1 | 5.70 |
| CHEMBL1908377 | PYRVINIUM PAMOATE | 4.0 | 1 | 5.47 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL866 | MYCOPHENOLIC ACID | EC50 | = | 180.0 | nM | 6.75 |
| CHEMBL1456 | MYCOPHENOLATE MOFETIL | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL400092 | LYCORINE | EC50 | = | 470.0 | nM | 6.33 |
| CHEMBL50588 | EMETINE | EC50 | = | 1430.0 | nM | 5.84 |
| CHEMBL5314365 | MONENSIN SODIUM | EC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1242 | PHENAZOPYRIDINE | EC50 | = | 2020.0 | nM | 5.70 |
| CHEMBL1908377 | PYRVINIUM PAMOATE | EC50 | = | 3350.0 | nM | 5.47 |