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Assay Detail

CHEMBL4726178

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of EGFR (unknown origin) expressed in baculovirus system using fluorescein labeled PDGFR-tide substrate peptide preincubated for 60 mins followed by ATP addition and measured after 60 mins by IMAP assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Epidermal growth factor receptor (CHEMBL203)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of quinoline-based irreversible BTK inhibitors.
de Bruin G,Demont D,de Zwart E,Verkaik S,Hoogenboom N,van de Kar B,van Lith B,Emmelot-van Hoek M,Gulrajani M,Covey T,Kaptein A,Barf T
Bioorg Med Chem Lett (2020) 30 : 127261 -127261
PubMed 32527559 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 18 7.45 8.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4779297 1 8.42
CHEMBL4791702 1 8.20
CHEMBL4798086 1 7.96
CHEMBL4794213 1 7.92
CHEMBL4763873 1 7.89
CHEMBL4744536 1 7.80
CHEMBL4759528 1 7.62
CHEMBL4755977 1 7.48
CHEMBL4796130 1 7.26
CHEMBL4792062 1 7.09
CHEMBL4745935 1 6.80
CHEMBL4752700 1 6.70
CHEMBL4756092 1 6.63
CHEMBL4787517 1 6.56
CHEMBL4800082 1 -
CHEMBL4743222 1 -
CHEMBL4791135 1 -
CHEMBL4782725 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4779297 IC50 = 3.8 nM 8.42
CHEMBL4791702 IC50 = 6.3 nM 8.20
CHEMBL4798086 IC50 = 11.0 nM 7.96
CHEMBL4794213 IC50 = 12.0 nM 7.92
CHEMBL4763873 IC50 = 13.0 nM 7.89
CHEMBL4744536 IC50 = 16.0 nM 7.80
CHEMBL4759528 IC50 = 24.0 nM 7.62
CHEMBL4755977 IC50 = 33.0 nM 7.48
CHEMBL4796130 IC50 = 55.0 nM 7.26
CHEMBL4792062 IC50 = 81.0 nM 7.09
CHEMBL4745935 IC50 = 159.0 nM 6.80
CHEMBL4752700 IC50 = 200.0 nM 6.70
CHEMBL4756092 IC50 = 233.0 nM 6.63
CHEMBL4787517 IC50 = 275.0 nM 6.56
CHEMBL4800082 IC50 > 1000.0 nM -
CHEMBL4743222 IC50 > 1000.0 nM -
CHEMBL4791135 IC50 > 1000.0 nM -
CHEMBL4782725 IC50 > 1000.0 nM -