Assay Detail
Binding
CHEMBL4732476
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Binding affinity to c-Myc G-quadruplex DNA (unknown origin) assessed as dissociation constant incubated for 5 mins by UV- vis spectrophotometric analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Not specified |
| Confidence | 3 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Benzimidazole-1,2,3-triazole hybrid molecules: synthesis and study of their interaction with G-quadruplex DNA
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 4.10 | 4.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4759761 | — | — | 1 | 4.10 |
| CHEMBL4786759 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4759761 | — | Kd | = | 79230.0 | nM | 4.10 |
| CHEMBL4786759 | — | Kd | = | 113000.0 | nM | - |